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Description Entry page for GPCR - 'OPIOID RECEPTORS_Kappa_Homo sapiens'
ClassCLASS A
FamilyOPIOID RECEPTORS
Sub-FamilyKappa
Cross References:
References
UniProtP41145 | Q499G4
EMBLU11053 | U17298 | L37362 | AF498922 | BC099912 | L36130 | U16860
InterProIPR000276 | IPR017452 | IPR000452 | IPR001418
PRODOM
GENEID4986
MIM165196
PRINTSPR00237 | PR00532 | PR00384
PFAMPF00001
Other GPCR resourcesGPCRDB | GPCR-OKB | GLIDA
Details:
Details
NameOPIOID RECEPTORS_Kappa_Homo sapiens
DescriptionRecName: Full=Kappa-type opioid receptor;AltName: Full=KOR-1
SpeciesHomo sapiens
Common NameHuman
NCBI Taxonomy9606
GeneOPRK1 | OPR
FunctionInhibits neurotransmitter release by reducing calciums ion currents and increasing potassium ion conductance
Fragment0
Sequence
MDSPIQIFRGEPGPTCAPSACLPPNSSAWFPGWAEPDSNGSAGSEDAQLEPAHISPAIPV
IITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTVYL
MNSWPFGDVLCKIVISIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINI
CIWLLSSSVGISAIVLGGTKVREDVDVIECSLQFPDDDYSWWDLFMKICVFIFAFVIPVL
IIIVCYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFVVCWTPIHIFILVEALG
STSHSTAALSSYYFCIALGYTNSSLNPILYAFLDENFKRCFRDFCFPLKMRMERQSTSRV
RNTVQDPAYLRDIDGMNKPV
Interacting with G-proteins:
G-proteins
NoNameCouplingPubMed
1Galpha-i1_Homo sapiensGi/o7624359
2Galpha-i3_Homo sapiensGi/o7624359
3Galpha-i2_Homo sapiensGi/o7624359
4Galpha-o_Homo sapiensGi/o7624359
5Galpha-z_Homo sapiensGi/o7624359
GPCR, G-protein, Effector interaction Visualizaton of GPCR, G-protein, Effector interaction at protein level